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Drug-Target Interaction

Drug

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PubChem ID:3038522
Structure:
Synonyms:
(4-(6-Methoxy-7-(3-piperidylpropoxy)quinazolin-4-yl)piperazinyl)-N-(4-(met
(4-(6-Methoxy-7-(3-piperidylpropoxy)quinazolin-4-yl)piperazinyl)-N-(4-(methylethoxy)phenyl)carboxamide
1-Piperazinecarboxamide, 4-(6-methoxy-7-(3-(1-piperidinyl)propoxy)-4-quinazolinyl)-N-(4-(1-methylethoxy)phenyl)-
387867-13-2
AC-1659
AC1MI50F
CHEMBL124660
CT 53518
CT-53518
CT53518
D06005
EC-000.2262
HMS3264G08
I14-1975
Kinome_3320
MLN 518
MLN-0518
MLN-518
MLN518, CT53518
NCGC00241097-01
NCGC00241097-02
NSC726292
S1043_Selleck
Tandutinib
Tandutinib (USAN/INN)
Tandutinib-Supplied by Selleck Chemicals
UNII-E1IO3ICJ9A

Target

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Uniprot ID:PIM1_HUMAN
Synonyms:
Proto-oncogene serine/threonine-protein kinase Pim-1
EC-Numbers:2.7.11.1
Organism:Homo sapiens
Human
PDB IDs:1XQZ 1XR1 1XWS 1YHS 1YI3 1YI4 1YWV 1YXS 1YXT 1YXU 1YXV 1YXX 2BIK 2BIL 2BZH 2BZI 2BZJ 2BZK 2C3I 2J2I 2O3P 2O63 2O64 2O65 2OBJ 2OI4 3BGP 3BGQ 3BGZ 3BWF 3C4E 3CXW 3CY2 3CY3 3DCV 3F2A
Structure:
3F2A

Binding Affinities:

Ki: Kd:Ic 50:Ec50/Ic50:
->10000--

References: