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Drug-Target Interaction

Drug

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PubChem ID:153999
Structure:
Synonyms:
(9S)-9-((Dimethylamino)methyl)-6,7,10,11-tetrahydro-9H,19H-5,21:12,17-dimethenodibenzo(e,k)pyrrolo(3,4-h)(1,4,13)oxadiazacyclohexadecene-18,20-dione
13-((Dimethylamino)methyl)-10,11,14,15-tetrahydro-4,9:16,21-dimetheno-1H,1
13-((Dimethylamino)methyl)-10,11,14,15-tetrahydro-4,9:16,21-dimetheno-1H,13H-dibenzo(e,k)pyrrolo(3,4-h)(1,4,13)oxadiazacyclohexadecene-1,3(2H)-dione
169939-94-0
1uu3
9H,18H-5,21:12,17-Dimethenodibenzo(e,k)pyrrolo(3,4-h)(1,4,13)oxadiazacyclohexadecine-18,20(19H)-dione, 9-((dimethylamino)methyl)-6,7,10,11-tetrahydro-, (9S)-
K00587a
LS-186984
LS-187626
LY 333531
LY-333,531
LY-333531
LY333531
LY4
Ruboxistaurin
Ruboxistaurin [INN]

Target

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Uniprot ID:KPCA_HUMAN
Synonyms:
PKC-A
PKC-alpha
Protein kinase C alpha type
EC-Numbers:2.7.11.13
Organism:Homo sapiens
Human
PDB IDs:2ELI
Structure:
2ELI

Binding Affinities:

Ki: Kd:Ic 50:Ec50/Ic50:
--360-

References: