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Drug-Target Interaction

Drug

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PubChem ID:127757
Structure:
Synonyms:
(S)-3-(8-((Dimethylamino)methyl)-6,7,8,9-tetrahydropyrido(1,2-a)indol-10-y
(S)-3-(8-((Dimethylamino)methyl)-6,7,8,9-tetrahydropyrido(1,2-a)indol-10-yl)-4-(1-methyl-1H-indol-3-yl)-1H-pyrrol-2,5-dione
(S)-3-(8-(Dimethylaminomethyl)-6,7,8,9-tetrahydropyrido(1,2-a)indol-10-yl)-4-(1-methyl-3-indolyl)-1H-pyrrole-2,5-dione hydrochloride
151342-35-7
1H-Pyrrol-2,5-dione, 3-(8-((dimethylamino)methyl)-6,7,8,9-tetrahydropyrido(1,2-a)indol-10-yl)-4-(1-methyl-1H-indol-3-yl)-, (S)-
1H-Pyrrole-2,5-dione, 3-(8-((dimethylamino)methyl)-6,7,8,9-tetrahydropyrido(1,2-a)indol-10-yl)-4-(1-methyl-1H-indol-3-yl)-, (S)-
C28H28N4O2.HCl
LS-173403
Ro 32-0432
Ro-32-0432

Target

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Uniprot ID:KPCA_HUMAN
Synonyms:
PKC-A
PKC-alpha
Protein kinase C alpha type
EC-Numbers:2.7.11.13
Organism:Homo sapiens
Human
PDB IDs:2ELI
Structure:
2ELI

Binding Affinities:

Ki: Kd:Ic 50:Ec50/Ic50:
--17.2-
--22-

References: